SCHEMBL115679

SCHEMBL115679

O=CC(N1CC=C(c2ccccc2-c2cnc(N3CCOCC3)nc2)CC1)n1ccc2cccnc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
CNR2 P34972 1/20 0.37
PDE9A O76083 1/20 0.34
AOC3 Q16853 10/20 0.34
KCNH2 Q12809 2/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
GLA P06280 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PIK3CA P42336 3/20 0.32
MTOR P42345 3/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113717 0.83 CNR2 (0.39) ALOX5APFEN1CNR2PDE9AAOC3
SCHEMBL114639 0.82 CNR2 (0.39) ALOX5APFEN1CNR2AOC3KCNH2
SCHEMBL113904 0.79 AOC3 (0.38) CNR2AOC3KCNH2
SCHEMBL115565 0.78 ALOX5AP (0.41) ALOX5APFEN1CNR2AOC3KCNH2
SCHEMBL3732871 0.76 NAMPT (0.44) AOC3
SCHEMBL113706 0.75 PTGS2 (0.33) FEN1CNR2MEN1ALDH1A1CASP1
SCHEMBL115691 0.71 SMN1; SMN2 (0.33) AOC3KCNH2MEN1ALDH1A1KMT2A
SCHEMBL113579 0.71 SMN1; SMN2 (0.33) AOC3KCNH2MEN1ALDH1A1KMT2A
SCHEMBL114774 0.70 LRRK2 (0.39) PIK3CAMTORPIK3CDPRKDC
SCHEMBL13039485 0.69 NAMPT (0.42) AOC3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed