SCHEMBL115565

SCHEMBL115565

Cc1cc(C)n(C(C=O)N2CC=C(c3ccccc3-c3cnc(N4CCOCC4)nc3)CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
CNR2 P34972 4/20 0.40
AOC3 Q16853 5/20 0.35
PRKAB2 O43741 1/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAG3 Q9UGI9 1/20 0.34
PRKAG2 Q9UGJ0 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
WDR5 P61964 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL112035 0.83 CNR2 (0.42) ALOX5APFEN1CNR2AOC3WDR5
SCHEMBL113179 0.81 CNR2 (0.40) ALOX5APFEN1CNR2AOC3WDR5
SCHEMBL115679 0.78 ALOX5AP (0.38) ALOX5APFEN1CNR2AOC3PIK3CD
SCHEMBL113998 0.77 AOC3 (0.39) ALOX5APFEN1CNR2AOC3WDR5
SCHEMBL3732875 0.76 CXCR3 (0.48) CNR2AOC3KCNH2
SCHEMBL113125 0.75 CXCR3 (0.40) ALOX5APFEN1CNR2AOC3KDM4E
SCHEMBL114041 0.74 CXCR3 (0.39) FEN1AOC3KDM4EKCNH2
SCHEMBL114405 0.74 CXCR3 (0.39) AOC3KCNH2
SCHEMBL113873 0.74 KDM4E (0.41) WDR5SMN1; SMN2KDM4E
SCHEMBL113141 0.74 CXCR3 (0.38) ALOX5APFEN1CNR2AOC3WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed