SCHEMBL11567937

SCHEMBL11567937

CCc1noc(N)c1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.43
LMNA P02545 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
GAA P10253 1/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 2/20 0.38
MLYCD O95822 1/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 6/20 0.37
RECQL P46063 1/20 0.37
HSD17B10 Q99714 6/20 0.36
ALDH1A1 P00352 3/20 0.36
POLB P06746 1/20 0.36
GLA P06280 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2334751 0.72
SCHEMBL11467892 0.72 LMNA (0.42) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL5157824 0.72
SCHEMBL2345949 0.70
SCHEMBL7222642 0.68
SCHEMBL9063960 0.68 MLYCD (0.37) CYP1A2CYP3A4CYP2C9CYP2C19MLYCD
SCHEMBL29172428 0.68 MAPK1 (0.37) KDM4ELMNACYP1A2CYP3A4CYP2C9
SCHEMBL13960108 0.66 CYP2A6 (0.41) KDM4ELMNAGAAMLYCDTP53
SCHEMBL11203252 0.64 GAA (0.38) KDM4EGAAHTTHPGDMAPK1
SCHEMBL8645691 0.64 PRKACA (0.43) KDM4EGAAHTTMAPK1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
EP-0002881-A1 5-Isoxazolylurea derivatives, their preparation, their use and compositions containing them FISONS plc (GB) 1979-07-11 EP disclosed