SCHEMBL11568629

SCHEMBL11568629

CC(C)C[C@H](N)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NC[C]=O

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.55
BACE2 Q9Y5Z0 4/20 0.55
PTPN1 P18031 3/20 0.53
IL1RN P18510 1/20 0.51
ERAP2 Q6P179 1/20 0.51
NPY4R P50391 6/20 0.50
NPY5R Q15761 5/20 0.50
NPY1R P25929 5/20 0.50
NPY2R P49146 3/20 0.49
OPRD1 P41143 2/20 0.48
OPRM1 P35372 1/20 0.48
OPRK1 P41145 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2195747 0.89 IL1RN (0.56) BACE1BACE2IL1RNERAP2NPY4R
SCHEMBL1372552 0.88 OPRD1 (0.56) BACE1BACE2OPRD1OPRM1OPRK1
SCHEMBL11566909 0.88 BACE1 (0.51) BACE1BACE2PTPN1IL1RNERAP2
SCHEMBL31696295 0.88 BACE1 (0.61) BACE1BACE2PTPN1IL1RNERAP2
SCHEMBL30123009 0.85 NAALAD2 (0.61) BACE1BACE2IL1RNERAP2NPY4R
SCHEMBL29973288 0.85 BACE1 (0.65) BACE1BACE2PTPN1NPY4RNPY1R
SCHEMBL31363027 0.85 OPRD1 (0.56) BACE1BACE2NPY4ROPRD1OPRM1
SCHEMBL6516934 0.84 BACE1 (0.57) BACE1BACE2PTPN1NPY4RNPY1R
SCHEMBL30798183 0.83 BACE1 (0.63) BACE1BACE2OPRD1
SCHEMBL29616324 0.82 BACE1 (0.58) BACE1BACE2PTPN1IL1RNERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4164571-A Medicament which antagonizes the action of gastrin and related polypeptides COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 1979-08-14 US claimed
US-4164571-A Medicament which antagonizes the action of gastrin and related polypeptides COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 1979-08-14 US disclosed