Prinomastat

Prinomastat

SCHEMBL115696

CC1(C)SCCN(S(=O)(=O)c2ccc(Oc3ccncc3)cc2)[C@H]1C(=O)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 20/20 1.00
MMP13 P45452 15/20 1.00
ADAM17 P78536 12/20 1.00
MMP3 P08254 10/20 1.00
MMP2 P08253 10/20 1.00
MMP9 P14780 10/20 1.00
MMP7 P09237 8/20 1.00
MMP8 P22894 6/20 1.00
MMP14 P50281 2/20 1.00
ADAM10 O14672 2/20 0.65
ADAM9 Q13443 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prinomastat SCHEMBL3955053 1.00 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL6801875 1.00 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL7765017 0.99 MMP1 (0.98) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL6810941 0.99 MMP1 (0.98) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL12272301 0.92 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6432297 0.90 MMP1 (0.81) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6336108 0.90 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6432301 0.90 MMP1 (0.81) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL3912779 0.90 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6344484 0.89 MMP1 (0.83) MMP1MMP13ADAM17MMP3MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 9215 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139320-A1 StarTrace: A Multiplex Drug Testing Platform for Personalized Medicine UNIV OF SOUTH CAROLINA (US) 2026-05-21 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12564575-B2 Early management, mitigation and prevention of sepsis and sepsis-like syndromes, including neo-natal ARDS due to infection, injury or iatrogenesis OPHIREX, INC (US) 2026-03-03 US claimed
US-12548678-B2 Methods and systems for machine learning analysis of single nucleotide polymorphisms in lupus AMPEL BIOSOLUTIONS, LLC (US) 2026-02-10 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20260007597-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRUS-INDUCED AIRWAY FIBROSIS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES (US) 2026-01-08 US claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US claimed
EP-4644418-A1 NANOBODY TARGETING BCMA, CHIMERIC ANTIGEN RECEPTOR AND USE THEREOF Hebei Senlang Biotechnology Co. Ltd. (CN) 2025-11-05 EP claimed
US-12383531-B2 PLA2 inhibitors for treatment of pathological conditions caused by hymenoptera envenomation, such as hemolysis, cerebral edema, and acute kidney injury OPHIREX, INC. (US) 2025-08-12 US claimed
US-20250221991-A1 COMBINATION THERAPY FOR THE TREATMENT OF CANCER METASTASES UNIVERSITY OF CINCINNATI (US) 2025-07-10 US claimed
US-20020147158-A1 Composition and method for preventing and treating sinusoidal obstruction syndrome and radiation-induced liver disease UNIVERSITY OF SOUTHERN CALIFORNIA 2002-10-10 US claimed
WO-2002067870-A2 COMPOSITION AND METHOD FOR PREVENTING AND TREATING SINUSOIDAL OBSTRUCTION SYNDROME AND RADIATION-INDUCED LIVER DISEASE UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2002-09-06 WO claimed
WO-2002059558-A2 MEANS AND METHODS FOR TREATMENT EVALUATION PRIMAGEN HOLDING B.V. (NL) 2002-08-01 WO claimed
EP-1225233-A2 Means and methods for treatment evaluation Amsterdam Support Diagnostics B.V. (NL) 2002-07-24 EP claimed
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP claimed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO claimed
EP-0935963-A2 The use of MMP-13 selective inhibitors for the treatment of osteoarthritis and other matrix metalloproteinase-mediated disorders Pfizer Products Inc. (US) 1999-08-18 EP claimed
EP-0874830-A1 METALLOPROTEINASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PHARMACEUTICAL USES, AND METHODS AND INTERMEDIATES USEFUL FOR THEIR PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 1998-11-04 EP claimed
US-5753653-A Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses AGOURON PHARMACEUTICALS, INC. (US) 1998-05-19 US claimed
WO-1997020824-A1 METALLOPROTEINASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PHARMACEUTICAL USES, AND METHODS AND INTERMEDIATES USEFUL FOR THEIR PREPARATION AGOURON PHARMACEUTICALS, INC. (US) 1997-06-12 WO claimed