Prinomastat

Prinomastat

SCHEMBL6801875

CC1(C)SCCN(S(=O)(=O)c2ccc(Oc3ccncc3)cc2)[C@@H]1C(=O)NO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 20/20 1.00
MMP13 P45452 15/20 1.00
ADAM17 P78536 12/20 1.00
MMP3 P08254 10/20 1.00
MMP2 P08253 10/20 1.00
MMP9 P14780 10/20 1.00
MMP7 P09237 8/20 1.00
MMP8 P22894 6/20 1.00
MMP14 P50281 2/20 1.00
ADAM10 O14672 2/20 0.65
ADAM9 Q13443 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prinomastat SCHEMBL3955053 1.00 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL115696 1.00 MMP1 (1.00) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL7765017 0.99 MMP1 (0.98) MMP1MMP13ADAM17MMP3MMP2
Prinomastat SCHEMBL6810941 0.99 MMP1 (0.98) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL12272301 0.92 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6432297 0.90 MMP1 (0.81) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6336108 0.90 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6432301 0.90 MMP1 (0.81) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL3912779 0.90 MMP1 (0.85) MMP1MMP13ADAM17MMP3MMP2
SCHEMBL6344484 0.89 MMP1 (0.83) MMP1MMP13ADAM17MMP3MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP claimed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO claimed
WO-1998047494-A2 NOVEL USE OF MATRIX METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1998-10-29 WO claimed
WO-2020252439-A1 CARBORANE HYDROXAMIC ACID MATRIX METALLOPROTEINASE AGENTS FOR BORON NEUTRON CAPTURE THERAPY LOYOLA UNIVERSITY OF CHICAGO (US) 2020-12-17 WO disclosed
CN-104174071-A COMPOSITIONS AND SYSTEMS FOR FORMING CROSSLINKED BIOMATERIALS AND ASSOCIATED METHODS OF PREPARATION AND USE ANGIODEVICE INTERNAT GMBH 2014-12-03 CN disclosed
US-20040229817-A1 Inhibitors of Hepatitis C virus, compositions and treatments using the same AGOURON PHARMACEUTICALS, INC. 2004-11-18 US disclosed
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP disclosed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO disclosed
WO-1998047494-A2 NOVEL USE OF MATRIX METALLOPROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 1998-10-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229817-A1 Inhibitors of Hepatitis C virus, compositions and treatments using the same TIMP3, MMP2, MMP7 MMP1 10/4885MMP13 6/4885ADAM17 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.