SCHEMBL11577256

SCHEMBL11577256

O=C1Cc2cc(Cl)ccc2Oc2ccc(Cl)cc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
AHR P35869 3/20 0.44
METAP1 P53582 1/20 0.41
NOTUM Q6P988 1/20 0.40
AR P10275 1/20 0.40
DRD2 P14416 2/20 0.39
DRD4 P21917 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
MAPT P10636 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TP53 P04637 1/20 0.39
CYP2C19 P33261 1/20 0.39
S100A4 P26447 1/20 0.38
KCNK2 O95069 1/20 0.38
ADRB2 P07550 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11577383 0.89 HRH4 (0.46) HPGDL3MBTL1AHRMETAP1NOTUM
SCHEMBL2375779 0.89 HPGD (0.52) HPGDL3MBTL1AHRNOTUMAR
SCHEMBL11564826 0.89 MAPK1 (0.47) HPGDL3MBTL1AHRMETAP1DRD2
SCHEMBL7112749 0.86 AR (0.41) HPGDL3MBTL1AHRMETAP1NOTUM
SCHEMBL7115732 0.82 MAPT (0.40) HPGDCYP3A4CYP2D6MAPTTP53
SCHEMBL1988800 0.82 CYP2C9 (0.45) HPGDL3MBTL1AHRNOTUMAR
SCHEMBL10463438 0.82 AHR (0.50) AHRMETAP1CYP1A2CYP3A4CYP2D6
SCHEMBL8817067 0.81 AHR (0.58) AHRMETAP1DRD2DRD4CYP1A2
SCHEMBL10646312 0.79 HRH4 (0.45) HPGDL3MBTL1AHRMETAP1NOTUM
SCHEMBL6287157 0.78 MAOA (0.54) AHRMETAP1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4118572-A CNS DEPRESSANTS, NEUROLEPTIC AGENTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-10-03 US disclosed
US-4105664-A Dibenz[b,f]oxepin derivatives HOFFMANN-LA ROCHE INC. (US) 1978-08-08 US disclosed
US-4100173-A DEPRESSANTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-07-11 US disclosed
US-4091023-A ANTISCHIZOPHRENIA AGENTS, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-05-23 US disclosed
US-4032525-A CNS DEPRESSANTS, NEUROLEPTICS HOFFMANN-LA ROCHE INC. (US) 1977-06-28 US disclosed