SCHEMBL11580468

SCHEMBL11580468

CS(=O)(=O)CCCN1C(=O)CN=C(c2ccccc2F)c2cc(Cl)ccc21

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 5/20 0.70
DRD3 P35462 2/20 0.70
KCNH2 Q12809 2/20 0.70
GHSR Q92847 2/20 0.70
HTR1A P08908 1/20 0.70
HTR3A P46098 1/20 0.70
TP53 P04637 5/20 0.55
LMNA P02545 3/20 0.50
NR1I2 O75469 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
OPRM1 P35372 1/20 0.50
CYP3A4 P08684 2/20 0.49
SLC22A1 O15245 1/20 0.49
ABCB11 O95342 1/20 0.49
PDE4D Q08499 1/20 0.49
GABRA1 P14867 4/20 0.48
GABRA5 P31644 4/20 0.48
GABRA3 P34903 4/20 0.48
GABRA2 P47869 4/20 0.48
GABRB2 P47870 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11579759 0.94 OPRK1 (0.72) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11578252 0.91 OPRK1 (0.72) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11581617 0.90 TP53 (0.63) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11580136 0.89 TP53 (0.56) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11579969 0.88 OPRK1 (0.69) OPRK1DRD3KCNH2GHSRHTR1A
Elfazepam SCHEMBL259108 0.87 OPRK1 (0.74) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11578526 0.87 OPRK1 (0.64) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11578262 0.86 OPRK1 (0.61) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11750221 0.86 OPRK1 (0.69) OPRK1DRD3KCNH2GHSRHTR1A
SCHEMBL11745535 0.86 OPRK1 (0.72) OPRK1DRD3KCNH2GHSRHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4079053-A Benzodiazepine derivatives SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1978-03-14 US disclosed
US-4010154-A Benzodiazepinones SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-03-01 US disclosed
US-3932637-A 1-ALKYLSULFONYLALKYL-1,4-BENZODIAZEPINONES SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1976-01-13 US disclosed