SCHEMBL1158441

SCHEMBL1158441

O=C1C=CC(=O)C(c2c[nH]c3ccccc23)=C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 1/20 0.60
PTPRF P10586 1/20 0.60
PTPN1 P18031 1/20 0.60
CDC25B P30305 1/20 0.60
SIRT2 Q8IXJ6 3/20 0.56
PRKCB P05771 2/20 0.56
PRKCA P17252 2/20 0.56
PRKD3 O94806 1/20 0.56
CCNB2 O95067 1/20 0.56
CCNE2 O96020 1/20 0.56
ABL1 P00519 1/20 0.56
PRKCG P05129 1/20 0.56
CDK1 P06493 1/20 0.56
PIM1 P11309 1/20 0.56
CDK4 P11802 1/20 0.56
CCNB1 P14635 1/20 0.56
PRKACA P17612 1/20 0.56
PRKACG P22612 1/20 0.56
PRKACB P22694 1/20 0.56
CCND1 P24385 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7951074 0.86 PTPN1 (0.73) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL27750430 0.78 PTPN11 (0.56) PTPRCPTPRFPTPN1CDC25BPRKCB
SCHEMBL27721368 0.78 PTPN11 (0.56) PTPN1NR4A2MEN1KMT2AALDH1A1
SCHEMBL21814328 0.78 LMNA (0.44) PTPRCPTPRFPTPN1CDC25BCCR6
SCHEMBL7737770 0.78 PDGFRB (0.44) PTPN1PRKD3CCNB2ABL1CDK1
SCHEMBL27771326 0.78 PTPN1 (0.61) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL27795880 0.78 PTPN1 (0.61) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL27771327 0.76 PTPRC (0.56) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL27771325 0.76 PTPRC (0.56) PTPRCPTPRFPTPN1CDC25BSIRT2
SCHEMBL9572016 0.75 PTPN1 (0.77) PTPRCPTPRFPTPN1CDC25BSIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 166 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111471046-B Carbazole indole quinone derivative and preparation method and application thereof 中国科学院成都有机化学有限公司 2024-04-05 CN claimed
CN-116924960-A Method for synthesizing 3-indolyl benzoquinone compound 郑州大学 2023-10-24 CN claimed
CN-113200967-B Indole benzoquinone compound, preparation method and application thereof 中国人民解放军陆军军医大学 2022-05-24 CN claimed
CN-113200967-A Indole benzoquinone compound, preparation method and application thereof 中国人民解放军陆军军医大学 2021-08-03 CN claimed
CN-112174872-A Indole benzoquinone derivative as fluorescent and photoacoustic imaging agent and application thereof 四川大学 2021-01-05 CN claimed
CN-110437124-A A kind of indoles quinone derivative and preparation method thereof CHENGDU ORGANIC CHEM CO LTD CAS 2019-11-12 CN claimed
CN-105646490-B The cyclohexadione compounds of indoles [1,2 a] pyrimidine [4,5 b] quinoline 7,13, preparation method and its medicinal usage 西北大学 2018-01-09 CN claimed
US-20080227168-A1 METHODS AND MATERIALS FOR EXTRA AND INTRACELLULAR DELIVERY OF CARBON NANOTUBES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2008-09-18 US claimed
EP-1900850-A1 PHOTOELECTROCHEMICAL METHOD OF SEPARATING WATER INTO HYDROGEN AND OXYGEN, USING MELANINS OR THE ANALOGUES, PRECURSORS OR DERIVATIVES THEREOF AS THE CENTRAL ELECTROLYSING ELEMENT Solis Herrera, Arturo (MX) 2008-03-19 EP claimed
EP-0959881-B1 SYNTHETIC METHODS FOR THE PREPARATION OF INDOLYLQUINONES AND MONO- AND BIS-INDOLYLQUINONES PREPARED THEREFROM SUGEN INC (US) 2005-09-21 EP claimed
US-20030060635-A1 Methods of using bis-indolylquinones TANG PENG C (US) 2003-03-27 US claimed
EP-0959881-A4 SYNTHETIC METHODS FOR THE PREPARATION OF INDOLYLQUINONES AND MONO- AND BIS-INDOLYLQUINONES PREPARED THEREFROM SUGEN INC (US) 2001-06-27 EP claimed
EP-0959881-A1 SYNTHETIC METHODS FOR THE PREPARATION OF INDOLYLQUINONES AND MONO- AND BIS-INDOLYLQUINONES PREPARED THEREFROM Sugen, Inc. (US) 1999-12-01 EP claimed
US-5786488-A DEHYDROBROMINATION OF A DIBROMOBENZOQUINONES WITH AT LEAST ONE INDOLES IN A POLAR SOLVENT AND A METAL CARBONATE TO FORM AN ANTITUMOR AGENT SUGEN, INC. (US) 1998-07-28 US claimed
WO-1998020874-A1 SYNTHETIC METHODS FOR THE PREPARATION OF INDOLYLQUINONES AND MONO- AND BIS-INDOLYLQUINONES PREPARED THEREFROM SUGEN, INC. (US) 1998-05-22 WO claimed
JP-57050959-A None JP disclosed
JP-57050959-A None JP disclosed
JP-S5750959-A INDOLE QUINONE COMPOUND YOSHITOMI PHARMACEUT IND LTD 1982-03-25 JP disclosed
JP-S5750959-A INDOLE QUINONE COMPOUND YOSHITOMI PHARMACEUT IND LTD 1982-03-25 JP disclosed
US-3987202-A METHOD OF TREATING PSORIASIS OKUN MILTON R 1976-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030060635-A1 Methods of using bis-indolylquinones IDO2, IDO1, IPO5 PTPRC 3030/4885PTPRF 3523/4885PTPN1 3612/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.