SCHEMBL11589058

SCHEMBL11589058

Cn1nc(-c2cccnc2)nc1-c1ccncc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.60
NR1H3 Q13133 2/20 0.60
NPC1 O15118 1/20 0.60
RAB9A P51151 1/20 0.60
HSD17B10 Q99714 2/20 0.48
HSD17B2 P37059 1/20 0.48
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4C Q9H3R0 1/20 0.46
CYP2A6 P11509 2/20 0.45
CYP2A13 Q16696 1/20 0.45
PPARA Q07869 3/20 0.45
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11592259 0.94 NR1H2 (0.60) NR1H2NR1H3NPC1RAB9AHSD17B10
SCHEMBL11589724 0.92 NR1H2 (0.61) NR1H2NR1H3NPC1RAB9AHSD17B10
SCHEMBL11588467 0.86 NR1H2 (0.72) NR1H2NR1H3NPC1RAB9AHSD17B10
SCHEMBL11590621 0.85 NR1H3 (0.83) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL11590519 0.85 NR1H3 (0.69) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL8405058 0.82 ALDH1A1 (0.50) NR1H2NR1H3NPC1RAB9AHSD17B10
SCHEMBL11311344 0.81 NR1H3 (0.71) NR1H2NR1H3NPC1RAB9AHSD17B2
SCHEMBL2365545 0.80 NR1H2 (0.62) NR1H2NR1H3NPC1RAB9AALDH1A1
SCHEMBL2313369 0.79 NR1H2 (0.54) NR1H2NR1H3NPC1RAB9AHSD17B10
SCHEMBL1460117 0.78 PPARA (0.50) NPC1RAB9AHSD17B10ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4111944-A SUBSTITUTED 1,2,4-TRIAZOLES MERCK & CO., INC. (US) 1978-09-05 US disclosed
US-3963731-A TREATMENT OF GOUT AND HYPERURICEMIA MERCK & CO., INC. (US) 1976-06-15 US disclosed
US-3947577-A 1,2,4-TRIAZOLES MERCK & CO., INC. (US) 1976-03-30 US disclosed