SCHEMBL11596174

SCHEMBL11596174

CCCCC(C)(C)C(=O)Nc1ncco1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.40
KDM4E B2RXH2 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
ACAT1 P24752 1/20 0.40
SOAT1 P35610 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
FFAR2 O15552 1/20 0.38
EPHX2 P34913 2/20 0.37
FAAH O00519 2/20 0.36
CES1 P23141 1/20 0.36
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21743428 0.78 KDM4E (0.45) KDM4ECYP3A4MAPTFFAR2EPHX2
SCHEMBL11544529 0.76 KDM4E (0.40) ARKDM4ETP53CYP3A4MAPT
SCHEMBL11595129 0.75 KDM4E (0.39) ARKDM4ETP53CYP3A4MAPT
SCHEMBL11536828 0.75 KDM4E (0.39) ARKDM4ETP53CYP3A4MAPT
SCHEMBL7091214 0.75 LMNA (0.50) EPHX2FAAHCES1
SCHEMBL11594989 0.74 KDM4E (0.38) ARKDM4ETP53CYP3A4MAPT
SCHEMBL11593235 0.73 KDM4E (0.38) ARKDM4ETP53CYP3A4MAPT
SCHEMBL11593210 0.73 ADORA1 (0.43)
SCHEMBL11594533 0.73 KMT2A (0.36) ARKMT2AFAAHCES1
SCHEMBL30846731 0.72 AR (0.56) ARKDM4ETP53CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4122183-A ANTIASTHMATIC LILLY INDUSTRIES LIMITED (GB) 1978-10-24 US disclosed