SCHEMBL11596389

SCHEMBL11596389

CC1(CC(=O)O)OCCc2c1[nH]c1ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.49
OGFRL1 Q5TC84 7/20 0.49
OPRL1 P41146 3/20 0.49
TSHR P16473 3/20 0.49
OPRD1 P41143 2/20 0.49
OPRK1 P41145 2/20 0.49
ALDH1A1 P00352 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
BLM P54132 1/20 0.49
PMP22 Q01453 1/20 0.49
SLC22A6 Q4U2R8 1/20 0.49
S1PR1 P21453 1/20 0.48
KDM4E B2RXH2 1/20 0.45
MAPT P10636 3/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11598173 0.89 OPRM1 (0.46) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11650527 0.88 OPRM1 (0.45) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11597100 0.88 OPRM1 (0.47) OPRM1OGFRL1OPRL1TSHROPRD1
Acetic Acid SCHEMBL11822954 0.88 OPRM1 (0.49) OPRM1OGFRL1OPRL1TSHROPRD1
Acetic Acid SCHEMBL11624482 0.88 OPRM1 (0.49) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11604174 0.87 OPRM1 (0.44) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11598201 0.87 OPRM1 (0.47) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11596132 0.87 OPRM1 (0.46) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11595954 0.87 OPRM1 (0.48) OPRM1OGFRL1OPRL1TSHROPRD1
SCHEMBL11598186 0.87 OPRM1 (0.49) OPRM1OGFRL1OPRL1TSHROPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3939178-A ANTIINFLAMMATORY, ANALGESIC, BACTERICIDE, FUNGICIDE AMERICAN HOME PRODUCTS CORPORATION (US) 1976-02-17 US claimed
US-4118394-A ANTIULCER, ANTIDEPRESSANT AYERST, MCKENNA & HARRISON LIMITED (CA) 1978-10-03 US disclosed
US-4076831-A Pyrano[3,4-b]-indole derivatives, pharmaceutical compositions and methods of use AMERICAN HOME PRODUCTS CORPORATION (US) 1978-02-28 US disclosed
US-4070371-A ANTIINFLAMMATORY, ANALGESIC, ANTIBACTERIAL, FUNGICIDES AMERICAN HOME PRODUCTS CORPORATION (US) 1978-01-24 US disclosed
US-4066780-A Pyranoindole derivatives as antiulcer agents AYERST MCKENNA AND HARRISON LTD. (CA) 1978-01-03 US disclosed
US-4066779-A ANTIDEPRESSANT, ANTIULCER AYERST, MCKENNA AND HARRISON LTD. (CA) 1978-01-03 US disclosed
US-4056538-A ANTIDEPRESSANTS, ANTIULCER AGENTS AYERST, MCKENNA & HARRISON LIMITED (CA) 1977-11-01 US disclosed
US-4056537-A CYCLIZATION, ACID CATALYST AYERST MCKENNA AND HARRISON LTD. (CA) 1977-11-01 US disclosed
US-4041169-A TREATING AND PREVENTING ULCERS AYERST MCKENNA AND HARRISON LTD. (CA) 1977-08-09 US disclosed
US-4012417-A ACID CATALYSTS AMERICAN HOME PRODUCTS CORPORATION (US) 1977-03-15 US disclosed
US-4003913-A ANTIDEPRESSANTS, ANTIULCER AGENTS AYERST MCKENNA AND HARRISON LTD. (CA) 1977-01-18 US disclosed
US-3974179-A ANTIINFLAMMATORY, ANALGESICS, BACTERICIDES, FUNGICIDES AMERICAN HOME PRODUCTS CORPORATION (US) 1976-08-10 US disclosed
US-3939178-A ANTIINFLAMMATORY, ANALGESIC, BACTERICIDE, FUNGICIDE AMERICAN HOME PRODUCTS CORPORATION (US) 1976-02-17 US disclosed