SCHEMBL11601080

SCHEMBL11601080

Cn1c(=O)n(C)c2cc(CC(N)C(=O)O)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 5/20 0.53
HSD17B10 Q99714 3/20 0.53
KDM4E B2RXH2 2/20 0.53
PTGS1 P23219 2/20 0.53
USP2 O75604 1/20 0.53
EGFR P00533 1/20 0.53
LCK P06239 1/20 0.53
FYN P06241 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
ALOX15 P16050 1/20 0.53
HTR2A P28223 1/20 0.53
PTGS2 P35354 1/20 0.53
RECQL P46063 1/20 0.53
HIF1A Q16665 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
TYR P14679 5/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
ALDH1A1 P00352 2/20 0.49
BRD4 O60885 1/20 0.49
BRPF1 P55201 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11599540 0.99 SLC7A5 (0.51) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL11706002 0.78 SLC7A5 (0.48) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL11600601 0.78 SLC7A5 (0.48) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL11601932 0.78 SLC7A5 (0.48) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL17229324 0.78 BRD4 (0.51) HSD17B10KDM4ESMN1; SMN2ALDH1A1BRD4
Hydrochloric Acid SCHEMBL11600341 0.77 SLC7A5 (0.47) SLC7A5HSD17B10KDM4EPTGS1USP2
Hydrochloric Acid SCHEMBL11602771 0.77 PKM (0.47) SLC7A5HSD17B10KDM4EPTGS1USP2
Hydrochloric Acid SCHEMBL11602211 0.77 SLC7A5 (0.47) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL28832116 0.77 SLC7A5 (0.43) SLC7A5HSD17B10KDM4EPTGS1USP2
SCHEMBL22862697 0.76 ALDH1A1 (0.65) HSD17B10KDM4EHIF1ATDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4073929-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1978-02-14 US disclosed
US-4069333-A 2-HYDRAZINO-3-PHENYLPROPIONIC ACID DECARBOXYLASE INHIBITORS, BENZOXAZOLE ANALINES MERCK & CO., INC. (US) 1978-01-17 US disclosed
US-4051251-A DECARBOXYLASE INHIBITOR, BENZIMIDAZOLE AND BENZOXAZOLE ALANINES N MERCK & CO., INC. (US) 1977-09-27 US disclosed