SCHEMBL1160657

SCHEMBL1160657

CCCC(=O)OC(=O)CCCCC(=O)O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.68
AKR1B1 P15121 1/20 0.58
GPR84 Q9NQS5 7/20 0.56
PPARG P37231 7/20 0.56
PPARD Q03181 7/20 0.56
PPARA Q07869 7/20 0.56
HDAC11 Q96DB2 5/20 0.56
TSHR P16473 5/20 0.56
PTPN1 P18031 3/20 0.56
TLR2 O60603 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
FABP4 P15090 2/20 0.56
KMT2A Q03164 2/20 0.56
SLC22A6 Q4U2R8 1/20 0.56
SLC22A8 Q8TCC7 1/20 0.56
MEN1 O00255 1/20 0.56
ESR1 P03372 1/20 0.56
ALOX15 P16050 1/20 0.56
PDE4A P27815 1/20 0.56
PDE3A Q14432 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14893175 0.98 ALDH1A1 (0.65) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL3518082 0.95 ALDH1A1 (0.68) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL3515582 0.91 AKR1B1 (0.65) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL27775207 0.91 AKR1B1 (0.73) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL195017 0.91 ALDH1A1 (0.83) ALDH1A1AKR1B1TSHRFFAR3HDAC3
Decanoic Acid SCHEMBL25428676 0.89 GPR84 (0.74) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL8574230 0.89 GPR84 (0.74) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL3515592 0.89 GPR84 (0.74) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL3516731 0.89 GPR84 (0.74) ALDH1A1AKR1B1GPR84PPARGPPARD
SCHEMBL7215249 0.89 GPR84 (0.74) ALDH1A1AKR1B1GPR84PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4066898-B1 BENZIMIDAZOLE COMPOUND OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDAL AND ACARICIDAL AGENT COMPRISING SAID COMPOUND, AND METHOD FOR USING SAID INSECTICIDAL AND ACARICIDAL AGENT NIHON NOHYAKU CO LTD (JP) 2026-01-07 EP disclosed
EP-4066898-A1 BENZIMIDAZOLE COMPOUND OR SALT THEREOF, AGRICULTURAL AND HORTICULTURAL INSECTICIDAL AND ACARICIDAL AGENT COMPRISING SAID COMPOUND, AND METHOD FOR USING SAID INSECTICIDAL AND ACARICIDAL AGENT Nihon Nohyaku Co., Ltd. (JP) 2022-10-05 EP disclosed
CN-109641696-A Vessel for preparing beverage 路易吉·拉瓦扎股份公司 2019-04-16 CN disclosed
CN-102742587-B Local topical administration formulations containing indoxacarb DU PONT 2014-06-25 CN disclosed
CN-101583278-B Local external application preparation containing indoxacarb DU PONT 2013-07-10 CN disclosed
CN-102742587-A Local topical administration formulations containing indoxacarb DU PONT 2012-10-24 CN disclosed
EP-2459569-A1 INSECTICIDAL 4-AMINO-THIENO[2,3-D]-PYRIMIDINE COMPOUNDS AND METHODS OF THEIR USE Merial Limited (US) 2012-06-06 EP disclosed
WO-2011014660-A1 INSECTICIDAL 4-AMINO-THIENO[2,3-D]-PYRIMIDINE COMPOUNDS AND METHODS OF THEIR USE MERIAL LIMITED (US) 2011-02-03 WO disclosed
CN-101854928-A The compositions that comprises avenanthramide CEAPRO INC 2010-10-06 CN disclosed
CN-101583278-A Local external application preparation containing indoxacarb DU PONT (US) 2009-11-18 CN disclosed
EP-0831088-B1 1,2,4-Triazine-3,5-dione derivatives as anticoccidial agents TAKEDA SCHERING PLOUGH ANIMAL (JP) 2002-11-27 EP disclosed
US-6294536-B1 CONTROL OF PROTOZOA AND REDUCTION IN THE INCIDENCE OF ASSOCIATED DISEASES AND DEATH AND CONSEQUENT IMPROVEMENT IN RETARDED GROWTH AND GENERAL CONDITION AND PREVENTING DECREASE GROWTH AND GENERAL CONDITION TAKEDA SCHERING-PLOUGH ANIMAL HEALTH K.K. (JP) 2001-09-25 US disclosed
CN-1054851-C 3-aryl-pyrone derivatives BAYER AG (DE) 2000-07-26 CN disclosed
US-5985875-A USEFUL AS ANTI-PROTOZOAL AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-16 US disclosed
CN-1215332-A Use of subsitituted aryl imidazoles BAYER AG (DE) 1999-04-28 CN disclosed
WO-1999011634-A1 TRIAZINE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-11 WO disclosed
EP-0831088-A1 1,2,4-Triazine-3,5-dione derivatives as anticoccidial agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-03-25 EP disclosed
CN-1085554-A 3-Arylpyrone Derivatives BAYER AG (DE) 1994-04-20 CN disclosed