SCHEMBL11615487

SCHEMBL11615487

COc1cc2c(CCNC(C)=O)c(C)[nH]c2cc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 1.00
MTNR1B P49286 15/20 1.00
CYP1A2 P05177 3/20 0.63
CYP3A4 P08684 3/20 0.63
CYP2D6 P10635 3/20 0.63
CYP2C9 P11712 2/20 0.63
CYP2C19 P33261 2/20 0.63
MEN1 O00255 1/20 0.63
LMNA P02545 1/20 0.63
NFKB1 P19838 1/20 0.63
MAPK1 P28482 1/20 0.63
SLC6A4 P31645 1/20 0.63
THPO P40225 1/20 0.63
HTR2B P41595 1/20 0.63
KMT2A Q03164 1/20 0.63
HIF1A Q16665 1/20 0.63
NQO2 P16083 4/20 0.54
SPR P35270 1/20 0.50
TSHR P16473 1/20 0.48
HSD17B10 Q99714 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8822777 0.88 MTNR1A (0.79) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7891030 0.86 MTNR1A (0.76) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7894816 0.86 MTNR1A (0.80) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL18239788 0.86 MTNR1A (0.75) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL16716178 0.85 MTNR1A (0.74) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL8822712 0.85 MTNR1A (0.74) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL15428065 0.84 MTNR1A (0.72) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL15427771 0.83 MTNR1A (0.71) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL677575 0.83 MTNR1A (1.00) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6
SCHEMBL7883115 0.80 MTNR1A (0.80) MTNR1AMTNR1BCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1047936-C Method for producing pharmaceutical composite containing alkylmelatonins LILLY CO ELI (US) 2000-01-05 CN disclosed
CN-1064807-A Preparation contains the method for the pharmaceutical composition of Alkylmelatonins LILLY CO ELI (US) 1992-09-30 CN disclosed
CN-1017426-B Process for preparing alkyl melatonin LILLY CO ELI (US) 1992-07-15 CN disclosed
CN-88100478-A alkyl melatonin 1988-08-17 CN disclosed
US-4087444-A Amides as ovulation inhibitors ELI LILLY AND COMPANY (US) 1978-05-02 US disclosed