SCHEMBL11617231

SCHEMBL11617231

CCC(C)COc1ccc(C2CCC(C#N)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
GRIA1 P42261 1/20 0.34
GRIA2 P42262 1/20 0.34
GRIA3 P42263 1/20 0.34
RAB9A P51151 1/20 0.34
GPR88 Q9GZN0 5/20 0.33
LTA4H P09960 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11616707 0.91 GPR88 (0.41) GPR88
SCHEMBL11522402 0.88 HRH3 (0.46) FFAR1SIGMAR1HRH3GRIA1GRIA2
SCHEMBL11522407 0.88 HRH3 (0.46) FFAR1SIGMAR1HRH3GRIA1GRIA2
SCHEMBL11619891 0.87 RAB9A (0.38) HRH3RAB9ALTA4H
SCHEMBL11615819 0.83 NQO1 (0.45) RAB9ALTA4HDRD2
SCHEMBL11036335 0.81 HRH3 (0.48) FFAR1SIGMAR1PDE4APDE4BPDE4C
SCHEMBL11617271 0.81 RAB9A (0.38) HRH3RAB9ADRD2
SCHEMBL11614025 0.81 ACACB (0.38) SIGMAR1HRH3GRIA1GRIA2GRIA3
SCHEMBL11619050 0.80 CYP1A2 (0.47) HRH3RAB9ALTA4HDRD2
SCHEMBL11523891 0.80 GRIA1 (0.44) HRH3GRIA1GRIA2GRIA3GPR88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4130502-A Liquid crystalline cyclohexane derivatives MERCK PATENT GESELLSCHAFT MIT (DE) 1978-12-19 US disclosed
US-4104274-A 1-Substituted-2-(2-pyridinyl)ethanone N-oxides WARNER-LAMBERT COMPANY (US) 1978-08-01 US disclosed
US-4076720-A 1-Substituted-2-(2-pyridinyl)ethanone N-oxides WARNER-LAMBERT COMPANY (US) 1978-02-28 US disclosed
US-4056619-A 1-Substituted-2-(2-pyridinyl)ethanone N-oxides WARNER-LAMBERT COMPANY (US) 1977-11-01 US disclosed