SCHEMBL11628784

SCHEMBL11628784

Cc1noc(C)c1CCC(=O)CCCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
GAA P10253 1/20 0.40
P2RX7 Q99572 2/20 0.39
ALDH1A1 P00352 5/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
TAS2R8 Q9NYW2 3/20 0.37
AR P10275 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL314801 0.87 MEN1 (0.45) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL12530346 0.80 P2RX7 (0.42) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL11631555 0.78 FFAR4 (0.41) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL12500526 0.76 P2RX7 (0.44) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL7033953 0.75 P2RX7 (0.46) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL314922 0.74 TDP1 (0.49) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL4182412 0.72 TDP1 (0.47) TDP1KMT2AMEN1GAAP2RX7
SCHEMBL14302719 0.72 P2RX7 (0.50) TDP1KMT2AMEN1P2RX7ALDH1A1
SCHEMBL2172793 0.72 P2RX7 (0.49) KMT2AMEN1GAAP2RX7ALDH1A1
SCHEMBL3690521 0.72 LMNA (0.41) TDP1KMT2AMEN1GAAP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4080334-A Intermediates in the total synthesis employing substituted isoxazole derivatives HOFFMANN-LA ROCHE INC. (US) 1978-03-21 US disclosed
US-4044004-A Total steroid synthesis employing substituted isoxazole derivatives HOFFMANN-LA ROCHE INC. (US) 1977-08-23 US disclosed
US-3985771-A Total steroid synthesis employing substituted isoxazole derivatives HOFFMANN-LA ROCHE INC. (US) 1976-10-12 US disclosed
US-3984427-A Preparation of vinyl lactones and corresponding Mannich bases HOFFMANN-LA ROCHE INC. (US) 1976-10-05 US disclosed
US-3984428-A Isoxazolyl-substituted perhydrobenzindenes HOFFMANN-LA ROCHE INC. (US) 1976-10-05 US disclosed