SCHEMBL11630673

SCHEMBL11630673

NC(=O)c1cnc(-c2ccccc2OCC2CC2)[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.47
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47
PDE4C Q08493 1/20 0.47
PDE4D Q08499 1/20 0.47
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
PARP1 P09874 1/20 0.40
IRAK4 Q9NWZ3 4/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
PARP15 Q460N3 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
BRD4 O60885 1/20 0.39
PDE1A P54750 2/20 0.38
PDE1B Q01064 2/20 0.38
PDE1C Q14123 2/20 0.38
MRGPRX1 Q96LB2 1/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11711842 0.90 PDE5A (0.48) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL11666115 0.89 IDO1 (0.51) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL11628709 0.85 KDM4E (0.51) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL11624906 0.83 GUSB (0.54) PDE5APDE1APDE1BPDE1CGUSB
SCHEMBL11629646 0.81 IDO1 (0.47) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7646746 0.81 PDE5A (0.41) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL9297225 0.81 PDE5A (0.55) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL11624834 0.81 PARP1 (0.56) PDE4APDE4BPDE4CPDE4DPARP1
SCHEMBL11624915 0.81 PDE5A (0.46) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL11626599 0.81 MEN1 (0.51) PDE5APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4082751-A ANTIALLERGENS BRISTOL-MYERS COMPANY (US) 1978-04-04 US disclosed