SCHEMBL11634008

SCHEMBL11634008

CSc1ccc2c(c1)N=C(N1CCN(CCO)CC1)c1cscc1N2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.53
CHRM1 P11229 7/20 0.43
HRH1 P35367 3/20 0.42
PAK1 Q13153 1/20 0.42
DRD2 P14416 8/20 0.40
DRD4 P21917 3/20 0.40
CHRM2 P08172 2/20 0.40
CHRM4 P08173 2/20 0.40
CHRM5 P08912 2/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
CHRM3 P20309 2/20 0.40
DRD1 P21728 2/20 0.40
ADRA1D P25100 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
ADRA1A P35348 2/20 0.40
ADRA1B P35368 2/20 0.40
HTR2B P41595 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11532011 0.89 CHRM1 (0.54) HRH4CHRM1HRH1PAK1DRD2
SCHEMBL11631525 0.85 HRH4 (0.74) HRH4CHRM1HRH1DRD2DRD4
SCHEMBL11637152 0.83 HRH4 (0.52) HRH4CHRM1HRH1PAK1DRD2
SCHEMBL11635638 0.83 HRH4 (0.62) HRH4CHRM1HRH1DRD2DRD4
SCHEMBL11631603 0.80 DRD2 (0.49) HRH4CHRM1HRH1PAK1DRD2
SCHEMBL11533334 0.77 HRH4 (0.54) HRH4CHRM1HRH1DRD2DRD4
SCHEMBL11632479 0.76 CHRM1 (0.71) HRH4CHRM1HRH1PAK1DRD2
SCHEMBL11622903 0.76 DRD4 (0.54) HRH4CHRM1HRH1DRD2DRD4
SCHEMBL11666986 0.74 CHRM1 (0.57) HRH4CHRM1HRH1PAK1DRD2
SCHEMBL11533730 0.73 CHRM1 (0.71) HRH4CHRM1HRH1PAK1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4087421-A NEUROLEPTIC, ANTI-DEPRESSANT AND ANALGESTIC ACTIVITY AMERICAN CYANAMID COMPANY (US) 1978-05-02 US disclosed
US-3951981-A NEUROLEPTIC, ANALGESIC AMERICAN CYANAMID COMPANY (US) 1976-04-20 US disclosed