SCHEMBL11634656

SCHEMBL11634656

O=C1CCC(c2cccc(O)c2Cl)=NN1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
PDE3A Q14432 9/20 0.38
PDE3B Q13370 8/20 0.38
PDE4B Q07343 4/20 0.38
PDE4A P27815 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
KCNH2 Q12809 1/20 0.38
PARP1 P09874 2/20 0.36
LMNA P02545 2/20 0.36
NPY1R P25929 1/20 0.36
NPY2R P49146 1/20 0.36
MAPT P10636 1/20 0.36
AXL P30530 1/20 0.36
TSHR P16473 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11637547 0.84 SMN1; SMN2 (0.51) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11657483 0.84 SMN1; SMN2 (0.59) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL9686080 0.82 SMN1; SMN2 (0.49) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11634644 0.78 PDE3A (0.47) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11626246 0.78 SMN1; SMN2 (0.59) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11738995 0.77 SMN1; SMN2 (0.46) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11738136 0.76 MEN1 (0.48) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11702816 0.75 SMN1; SMN2 (0.42) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11702077 0.74 SMN1; SMN2 (0.54) SMN1; SMN2PDE3APDE3BPDE4BPDE4A
SCHEMBL11743380 0.74 SMN1; SMN2 (0.43) SMN1; SMN2PDE3APDE3BPDE4BPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4082843-A 3-(3-(3-Substituted amino-2-hydroxypropoxy)phenyl)-6-hydrazino pyridazines and their use as vasodilators and β-adrenergic blocking agents SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1978-04-04 US disclosed