SCHEMBL1163671

SCHEMBL1163671

CCOC(=O)[C@@H](NC(=O)OC(C)(C)C)C1CC2CCC(C1)N2C(=O)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.49
CHRM1 P11229 7/20 0.45
CHRM4 P08173 1/20 0.45
CHRM5 P08912 1/20 0.45
SYK P43405 1/20 0.45
KLK7 P49862 4/20 0.44
KLK5 Q9Y337 3/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
AGTR2 P50052 1/20 0.42
HTR2C P28335 1/20 0.40
PPARA Q07869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3744365 0.92 CTSL (0.50) CTSLSYKKLK7KLK5KMT2A
SCHEMBL3748764 0.92 CTSL (0.50) CTSLSYKKLK7KLK5KMT2A
SCHEMBL6880634 0.91 CTSL (0.51) CTSLSYKKLK7KLK5KMT2A
SCHEMBL11902313 0.91 CTSL (0.51) CTSLSYKKLK7KLK5KMT2A
SCHEMBL16120917 0.84 CTSL (0.49) CTSLSYKKLK7KLK5PPARA
SCHEMBL1163483 0.83 CYP3A4 (0.47) CHRM1CHRM4CHRM5KMT2AHTR2C
SCHEMBL21653773 0.83 KMT2A (0.62) CTSLCHRM1CHRM4CHRM5SYK
SCHEMBL21653658 0.83 KMT2A (0.62) CTSLCHRM1CHRM4CHRM5SYK
SCHEMBL21653776 0.83 KMT2A (0.62) CTSLCHRM1CHRM4CHRM5SYK
SCHEMBL7489001 0.83 KMT2A (0.62) CTSLCHRM1CHRM4CHRM5SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011018796-A1 AN IMPROVED PROCESS FOR THE SYNTHESIS OF ALKYL/ARALKYL (2S)-2-(TERT-BUTOXYCARBONYL)-AMINO-2-[-8-AZABICYCLO[3.2.1]OCT-3-YL]-EXO-ACETATE AND ANALOGS THEREOF: KEY INTERMEDIATES FOR THE PREPARATION OF DPPIV INHIBITORS LUPIN LIMITED (IN) 2011-02-17 WO disclosed