SCHEMBL1163483

SCHEMBL1163483

COC(=O)[C@@H](NC(=O)OCc1ccccc1)C1CC2CCC(C1)N2C(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.47
TSHR P16473 7/20 0.47
ALDH1A1 P00352 6/20 0.47
CYP2C9 P11712 4/20 0.47
CYP2C19 P33261 4/20 0.47
CYP1A2 P05177 4/20 0.47
POLB P06746 1/20 0.47
CYP2D6 P10635 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HTR2C P28335 1/20 0.46
TRPM8 Q7Z2W7 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11901994 0.91 ALDH1A1 (0.46) CYP3A4TSHRALDH1A1CYP2C9CYP2C19
SCHEMBL3748764 0.91 CTSL (0.50) SMN1; SMN2KMT2AHTR2CNPC1RAB9A
SCHEMBL3744365 0.91 CTSL (0.50) SMN1; SMN2KMT2AHTR2CNPC1RAB9A
SCHEMBL11965223 0.87 HTR2C (0.47) CYP3A4TSHRALDH1A1CYP2C9CYP2C19
SCHEMBL3748271 0.85 SMN1; SMN2 (0.48) CYP2C19SMN1; SMN2HTR2CNPC1RAB9A
SCHEMBL3746212 0.85 SMN1; SMN2 (0.48) CYP2C19SMN1; SMN2HTR2CNPC1RAB9A
SCHEMBL11965219 0.85 HTR2C (0.50) CYP3A4TSHRALDH1A1CYP2C9CYP2C19
SCHEMBL1163564 0.84 CTSL (0.41) CYP3A4TSHRALDH1A1CYP2C9CYP2C19
SCHEMBL11965235 0.83 HTR2C (0.42) POLBSMN1; SMN2LMNAMEN1KMT2A
SCHEMBL11902313 0.83 CTSL (0.51) KMT2AMAPK1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011018796-A1 AN IMPROVED PROCESS FOR THE SYNTHESIS OF ALKYL/ARALKYL (2S)-2-(TERT-BUTOXYCARBONYL)-AMINO-2-[-8-AZABICYCLO[3.2.1]OCT-3-YL]-EXO-ACETATE AND ANALOGS THEREOF: KEY INTERMEDIATES FOR THE PREPARATION OF DPPIV INHIBITORS LUPIN LIMITED (IN) 2011-02-17 WO disclosed