SCHEMBL11640552

SCHEMBL11640552

CN(C)CCCN1C(=O)C(C)(C)c2ccccc21

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.78
CYP1A2 P05177 3/20 0.78
KMT2A Q03164 3/20 0.78
LMNA P02545 6/20 0.50
HRH1 P35367 5/20 0.50
MAPT P10636 5/20 0.50
TP53 P04637 5/20 0.50
HTR1A P08908 4/20 0.50
DRD2 P14416 4/20 0.50
HTR2A P28223 4/20 0.50
SLC6A4 P31645 4/20 0.50
HTR6 P50406 4/20 0.50
SLC22A1 O15245 3/20 0.50
CHRM2 P08172 3/20 0.50
CHRM4 P08173 3/20 0.50
CHRM5 P08912 3/20 0.50
CHRM1 P11229 3/20 0.50
ADRA2B P18089 3/20 0.50
ADRA2C P18825 3/20 0.50
CHRM3 P20309 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11640659 0.91 KMT2A (0.63) CYP2D6CYP1A2KMT2ALMNAHRH1
Dimetacrine SCHEMBL29578094 0.88 CYP2D6 (1.00) CYP2D6CYP1A2KMT2ALMNAHRH1
Dimetacrine SCHEMBL50120 0.88 CYP2D6 (1.00) CYP2D6CYP1A2KMT2ALMNAHRH1
SCHEMBL11639312 0.83 KMT2A (0.57) CYP2D6CYP1A2KMT2ALMNAHRH1
SCHEMBL507636 0.82 KMT2A (0.51) CYP2D6CYP1A2KMT2ALMNAMAPT
SCHEMBL319784 0.82 KMT2A (0.51) CYP2D6CYP1A2KMT2ALMNAMAPT
SCHEMBL11640444 0.81 CYP2D6 (0.58) CYP2D6CYP1A2KMT2ALMNAHRH1
SCHEMBL11639729 0.80 CYP2D6 (0.57) CYP2D6CYP1A2KMT2ALMNAHRH1
SCHEMBL23865489 0.80 TP53 (0.50) CYP2D6CYP1A2KMT2ALMNAMAPT
SCHEMBL507840 0.79 CYP1A2 (0.49) CYP2D6CYP1A2KMT2ALMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4123543-A ANTIDEPRESSANTS AB KABI (SE) 1978-10-31 US disclosed
US-4117144-A ANTIDEPRESSANTS AB KABI (SE) 1978-09-26 US disclosed
US-3947451-A TREATMENT OF PSYCHIATRIC AND PSYCHOSOMATIC DISEASES AB KABI (SW) 1976-03-30 US disclosed