SCHEMBL11645644

SCHEMBL11645644

COc1cccc(Oc2cccc(NC(=O)C(C)N)c2)c1

nearest known ligand 0.65

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 6/20 0.65
TSHR P16473 2/20 0.61
ALDH1A1 P00352 2/20 0.61
L3MBTL1 Q9Y468 1/20 0.55
MTNR1A P48039 2/20 0.55
TP53 P04637 2/20 0.54
RXFP1 Q9HBX9 1/20 0.54
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
KMT2A Q03164 2/20 0.52
NLRP3 Q96P20 1/20 0.52
PKM P14618 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
THRB P10828 1/20 0.52
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11642716 0.93 MTNR1B (0.64) MTNR1BTSHRALDH1A1L3MBTL1MTNR1A
SCHEMBL1980614 0.90 MTNR1B (0.80) MTNR1BTSHRALDH1A1MTNR1ATP53
SCHEMBL11637763 0.90 MTNR1B (0.80) MTNR1BTSHRALDH1A1MTNR1ATP53
SCHEMBL11645434 0.89 XIAP (0.58) MTNR1BTSHRALDH1A1NPC1RAB9A
SCHEMBL11645837 0.86 CDK8 (0.53) MTNR1BTSHRALDH1A1KMT2ASMN1; SMN2
SCHEMBL11645404 0.85 MTNR1B (0.63) MTNR1BTSHRALDH1A1MTNR1ANPC1
SCHEMBL11646067 0.85 XIAP (0.54) MTNR1BTSHRALDH1A1TP53NPC1
SCHEMBL11644195 0.85 XIAP (0.48) MTNR1BTSHRALDH1A1RAB9AKMT2A
SCHEMBL11645013 0.85 XIAP (0.54) MTNR1BTSHRALDH1A1L3MBTL1NPC1
SCHEMBL11641056 0.84 MTNR1B (0.60) MTNR1BTSHRALDH1A1MTNR1ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4088780-A ANTHELMINTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1978-05-09 US disclosed
US-4032655-A PHENYLGUANIDINES USEFUL AS ANTHELMINTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1977-06-28 US disclosed
US-4024176-A Substituted phenylguanidines and processes for their preparation and use BAYER AKTIENGESELLSCHAFT (DT) 1977-05-17 US disclosed
US-3993682-A Substituted phenylguanidines and processes for their preparation and use BAYER AKTIENGESELLSCHAFT (DT) 1976-11-23 US disclosed