SCHEMBL11646754

SCHEMBL11646754

CC(N)C(=O)Nc1ccc(S(=O)(=O)c2ccc(Br)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.53
CA2 P00918 10/20 0.53
CA12 O43570 4/20 0.53
CA9 Q16790 4/20 0.53
TAAR1 Q96RJ0 2/20 0.53
CA7 P43166 6/20 0.50
CA14 Q9ULX7 6/20 0.50
PKM P14618 2/20 0.49
CYP2C19 P33261 1/20 0.49
ATM Q13315 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
IDO1 P14902 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
S1PR3 Q99500 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748983 0.89 TAAR1 (0.64) TAAR1ALDH1A1MAPTMEN1KMT2A
SCHEMBL11664191 0.86 SMN1; SMN2 (0.64) CA1CA2CA12CA9ALDH1A1
SCHEMBL11644202 0.86 PKM (0.64) CA1CA2CA12CA9TAAR1
SCHEMBL11642546 0.86 PKM (0.67) CA1CA2CA12CA9TAAR1
SCHEMBL11640068 0.86 TAAR1 (0.67) CA1CA2CA12CA9TAAR1
SCHEMBL11646738 0.85 CA1 (0.58) CA1CA2CA12CA9TAAR1
SCHEMBL11642552 0.84 CA1 (0.51) CA1CA2CA12CA9TAAR1
SCHEMBL11643956 0.84 KMT2A (0.59) CA1CA2CA12CA9TAAR1
SCHEMBL11641981 0.82 PKM (0.51) CA1CA2CA12CA9TAAR1
SCHEMBL11645058 0.82 LMNA (0.55) CA1CA2CA12CA9TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4088780-A ANTHELMINTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1978-05-09 US disclosed
US-4032655-A PHENYLGUANIDINES USEFUL AS ANTHELMINTIC AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1977-06-28 US disclosed
US-4024176-A Substituted phenylguanidines and processes for their preparation and use BAYER AKTIENGESELLSCHAFT (DT) 1977-05-17 US disclosed
US-3993682-A Substituted phenylguanidines and processes for their preparation and use BAYER AKTIENGESELLSCHAFT (DT) 1976-11-23 US disclosed