SCHEMBL11665017

SCHEMBL11665017

C=CCn1c(=O)c2[nH]cnc2n(CC(C)CC)c1=O

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 14/20 0.72
ADORA2A P29274 12/20 0.72
PDE4A P27815 11/20 0.72
PDE4B Q07343 11/20 0.72
PDE4C Q08493 11/20 0.72
PDE4D Q08499 11/20 0.72
PDE2A O00408 2/20 0.55
PDE1A P54750 2/20 0.55
PDE1B Q01064 2/20 0.55
PDE1C Q14123 2/20 0.55
CFTR P13569 2/20 0.52
PDE5A O76074 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
ADORA1 P30542 1/20 0.52
SCN1A P35498 1/20 0.52
PDE6C P51160 1/20 0.52
PDE3B Q13370 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11073850 0.89 ADORA2B (0.78) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10339736 0.86 ADORA2A (0.74) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL516503 0.85 ADORA2B (1.00) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL9429985 0.81 PDE4A (0.85) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL7597430 0.77 ADORA2B (0.82) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL4623640 0.76 ADORA2A (0.76) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL5405285 0.76 ADORA2A (0.86) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10013824 0.74 CYP3A4 (0.59) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL10013807 0.74 CYP3A4 (0.59) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL8350764 0.72 PDE4A (0.77) ADORA2BADORA2APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4089959-A Long-acting xanthine bronchodilators and antiallergy agents COOPER LABORATORIES, INC. (US) 1978-05-16 US disclosed