SCHEMBL9429985

SCHEMBL9429985

C=CCn1c(=O)c2[nH]cnc2n(CCCC)c1=O

nearest known ligand 0.85

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.85
PDE4B Q07343 14/20 0.85
PDE4C Q08493 14/20 0.85
PDE4D Q08499 14/20 0.85
ADORA2A P29274 12/20 0.85
ADORA2B P29275 11/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL516503 0.88 ADORA2B (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3186630 0.88 PDE4A (0.94) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL11361392 0.86 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3842077 0.85 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381259 0.85 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381240 0.85 ADORA2B (0.94) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3190853 0.85 ADORA2B (0.92) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381263 0.84 ADORA2B (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381253 0.84 ADORA2B (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7744388 0.84 ADORA2B (0.97) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4469698-A SEDATIVES, TRANQUILIZERS SOCIETE D'ASSISTANCE TECHNIQUE POUR PRODUITS NESTLE S.A. (CH) 1984-09-04 US claimed
US-5338741-A Cardiotonic agents NESTEC S.A. (CH) 1994-08-16 US disclosed
EP-0269841-B1 1-HYDROXYALKYL XANTHINES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM SOCIETE DES PRODUITS NESTLE S.A. (CH) 1992-11-11 EP disclosed
US-5053433-A Photodiesterase inhibitor SOCIETE ANONYME DITE: L'OREAL (FR) 1991-10-01 US disclosed
EP-0269841-A1 1-Hydroxyalkyl xanthines, processes for their preparation and medicaments containing them SOCIETE DES PRODUITS NESTLE S.A. (CH) 1988-06-08 EP disclosed