SCHEMBL11670367

SCHEMBL11670367

CCOC(=O)C1=C(N)NC(N)=C(C(=O)OCC)C1c1cccc2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.59
NPSR1 Q6W5P4 2/20 0.59
PKM P14618 1/20 0.56
KMT2A Q03164 6/20 0.49
MEN1 O00255 5/20 0.49
CYP2C9 P11712 3/20 0.49
KDM4E B2RXH2 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2C19 P33261 2/20 0.49
HIF1A Q16665 2/20 0.49
HSD17B10 Q99714 2/20 0.49
GAA P10253 2/20 0.49
ALDH1A1 P00352 2/20 0.49
TSHR P16473 2/20 0.49
HPGD P15428 1/20 0.49
TP53 P04637 1/20 0.49
CYP2D6 P10635 1/20 0.49
NFKB1 P19838 1/20 0.49
THPO P40225 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11522544 0.94 MAPT (0.65) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL2996737 0.88 MAPT (0.70) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL11829270 0.84 CYP2C9 (0.67) MAPTNPSR1KMT2AMEN1CYP2C9
SCHEMBL11804731 0.84 MAPT (0.65) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL11669240 0.83 CA1 (0.55) MAPTNPSR1KMT2AMEN1CYP2C9
SCHEMBL11693805 0.82 ALDH1A1 (0.58) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL2991073 0.82 PKM (0.69) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL11781375 0.81 MAPT (0.52) MAPTNPSR1PKMKMT2AMEN1
SCHEMBL11669776 0.81 ALDH1A1 (0.51) MAPTNPSR1KMT2AMEN1CYP2C9
SCHEMBL11829351 0.81 NPSR1 (0.64) MAPTNPSR1PKMKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3957998-A ADMINISTERING BAYER AKTIENGESELLSCHAFT (DT) 1976-05-18 US claimed
US-4049662-A HYPOTENSIVE AGENTS, VASODILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-09-20 US disclosed
US-4016277-A ANTIHYPERTENSIVE AGENTS AND CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-04-05 US disclosed
US-3988458-A HYPOTENSIVE, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-10-26 US disclosed
US-3959474-A 2,6-Diamino-1,4-dihydropyridine-3,5-dicarboxylic acid esters used as coronary vessel dilators and anti-hypertensive agents BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed
US-3957998-A ADMINISTERING BAYER AKTIENGESELLSCHAFT (DT) 1976-05-18 US disclosed
US-3950336-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-13 US disclosed