Benderizine

Benderizine

SCHEMBL11673167

COc1ccc(CC2(C)CN(C(c3ccccc3)c3ccccc3)CCN2C)cc1OC

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KMT2A Q03164 2/20 0.45
POLB P06746 2/20 0.42
MEN1 O00255 1/20 0.42
EBP Q15125 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
DRD3 P35462 2/20 0.41
TMEM97 Q5BJF2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CACNA2D1 P54289 1/20 0.41
CACNA1B Q00975 1/20 0.41
CACNB1 Q02641 1/20 0.41
CACNA1C Q13936 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benderizine SCHEMBL1816506 1.00 ALDH1A1 (0.47) ALDH1A1GAATDP1KMT2APOLB
Benderizine SCHEMBL11673215 0.99 ALDH1A1 (0.46) ALDH1A1GAATDP1KMT2APOLB
SCHEMBL11628159 0.94 ACHE (0.43) ALDH1A1GAATDP1KMT2APOLB
Hydrochloric Acid SCHEMBL11630062 0.93 ACHE (0.42) ALDH1A1GAATDP1KMT2APOLB
Hydrochloric Acid SCHEMBL11672394 0.93 RECQL (0.47) ALDH1A1GAATDP1KMT2AMEN1
Benderizine SCHEMBL11673362 0.92 ALDH1A1 (0.43) ALDH1A1GAATDP1KMT2APOLB
SCHEMBL11630816 0.90 GAA (0.44) ALDH1A1GAATDP1KMT2AMEN1
SCHEMBL11630162 0.90 ALDH1A1 (0.42) ALDH1A1GAATDP1KMT2AMEN1
SCHEMBL11628858 0.89 ACHE (0.46) ALDH1A1GAATDP1KMT2APOLB
Hydrochloric Acid SCHEMBL11630911 0.88 ACHE (0.45) KMT2APOLBMEN1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3996360-A ANTIARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1976-12-07 US claimed
US-4031216-A CARDIAC DISEASE, ARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1977-06-21 US disclosed
US-3996360-A ANTIARRHYTHMIA KNOLL A.G. CHEMISCHE FABRIKEN (DT) 1976-12-07 US disclosed