SCHEMBL1167350

SCHEMBL1167350

CC(=O)CCCCn1cc(NC(=O)c2nc(C)sc2-c2ccccc2)cn1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
RAB9A P51151 1/20 0.46
HCRTR2 O43614 14/20 0.45
POLB P06746 1/20 0.44
HCRTR1 O43613 3/20 0.44
ITK Q08881 1/20 0.41
SCD O00767 1/20 0.41
SCD5 Q86SK9 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1167565 0.79 HCRTR2 (0.60) ALDH1A1HCRTR2POLBHCRTR1ITK
SCHEMBL1167055 0.78 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL1166697 0.74 HCRTR2 (0.61) HCRTR2HCRTR1
SCHEMBL1166840 0.72 HCRTR2 (0.51) HCRTR2HCRTR1
SCHEMBL1167197 0.72 HCRTR2 (0.45) ALDH1A1HCRTR2HCRTR1
SCHEMBL1166320 0.72 KDM4E (0.45) ALDH1A1MAPTHCRTR2HCRTR1ITK
SCHEMBL1167087 0.71 HCRTR2 (0.70) ALDH1A1HCRTR2POLBHCRTR1SMN1; SMN2
SCHEMBL1166791 0.70 CYP1A2 (0.51) ALDH1A1MAPTRAB9APOLBSMN1; SMN2
SCHEMBL1166403 0.69 FPR2 (0.44) ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL1166775 0.69 LPAR1 (0.49) ALDH1A1MAPTPOLBSCDSCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110034516-A1 AMINOPYRAZOLE DERIVATIVES ACTELION (CH) 2011-02-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034516-A1 AMINOPYRAZOLE DERIVATIVES CYP3A43, CYP1A2, CYP3A5 ALDH1A1 96/4885MAPT 2198/4885RAB9A 1767/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.