SCHEMBL1167197

SCHEMBL1167197

CC(=O)CCCCn1cc(NC(=O)c2nc(C)oc2-c2ccc(Cl)cc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.45
HCRTR1 O43613 3/20 0.45
ALDH1A1 P00352 1/20 0.41
HDAC3 O15379 2/20 0.40
JAK2 O60674 2/20 0.40
JAK1 P23458 2/20 0.40
TYK2 P29597 2/20 0.40
JAK3 P52333 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
HPGD P15428 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1166697 0.85 HCRTR2 (0.61) HCRTR2HCRTR1
SCHEMBL1166534 0.77 HCRTR2 (0.51) HCRTR2HCRTR1ALDH1A1
SCHEMBL1166513 0.76 HCRTR2 (0.53) HCRTR2HCRTR1
SCHEMBL1167055 0.74 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL1166786 0.73 HCRTR2 (0.62) HCRTR2HCRTR1ALDH1A1HPGDKDM4E
SCHEMBL1167892 0.73 HCRTR2 (0.68) HCRTR2HCRTR1
SCHEMBL1166629 0.73 HCRTR2 (0.58) HCRTR2HCRTR1
SCHEMBL1167350 0.72 ALDH1A1 (0.46) HCRTR2HCRTR1ALDH1A1
SCHEMBL1166992 0.72 HCRTR2 (0.64) HCRTR2HCRTR1ALDH1A1
SCHEMBL1166316 0.71 HDAC3 (0.45) ALDH1A1HDAC3JAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110034516-A1 AMINOPYRAZOLE DERIVATIVES ACTELION (CH) 2011-02-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110034516-A1 AMINOPYRAZOLE DERIVATIVES CYP3A43, CYP1A2, CYP3A5 HCRTR2 2700/4885HCRTR1 2862/4885ALDH1A1 96/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.