SCHEMBL11679644

SCHEMBL11679644

COC(=O)C(C)c1ccc2c(c1)Cc1cc(OC)ccc1-2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
PTGS2 P35354 5/20 0.48
PTGS1 P23219 2/20 0.48
AKR1C3 P42330 2/20 0.48
AKR1C2 P52895 2/20 0.48
TSHR P16473 2/20 0.48
CDC42 P60953 1/20 0.48
RAC1 P63000 1/20 0.48
CYP1A2 P05177 1/20 0.48
SLC22A6 Q4U2R8 1/20 0.48
MAPT P10636 2/20 0.46
LMNA P02545 1/20 0.46
CYP2C9 P11712 1/20 0.46
METAP1 P53582 1/20 0.46
APP P05067 1/20 0.44
CYP2C19 P33261 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11682544 0.87 AKR1C3 (0.64) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL11682946 0.83 RAB9A (0.44) TDP1L3MBTL1PTGS2PTGS1MAPT
SCHEMBL8754690 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL505811 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL29508603 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL505819 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL29403959 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL505799 0.79 TDP1 (0.77) TDP1L3MBTL1PTGS2PTGS1AKR1C3
SCHEMBL11681428 0.79 TLR9 (0.51) AKR1C3AKR1C2MAPTLMNA
SCHEMBL4007061 0.77 MEN1 (0.54) TDP1L3MBTL1PTGS2PTGS1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4052436-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1977-10-04 US disclosed
US-3989841-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1976-11-02 US disclosed