SCHEMBL11683042

SCHEMBL11683042

Nc1nnc(SC2CCCCC2)s1

nearest known ligand 0.96

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.96
FBP1 P09467 1/20 0.48
POLB P06746 2/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 5/20 0.41
HPGD P15428 4/20 0.40
ATM Q13315 1/20 0.40
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
GFER P55789 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12949443 0.77 SMN1; SMN2 (0.59) SMN1; SMN2GAAALDH1A1HPGDMAPT
SCHEMBL31715322 0.75 SMN1; SMN2 (0.62) SMN1; SMN2FBP1ALDH1A1HPGDATM
SCHEMBL11723394 0.73 SMN1; SMN2 (0.54) SMN1; SMN2ALDH1A1HPGDMAPTHTT
SCHEMBL30106080 0.72 SMN1; SMN2 (0.57) SMN1; SMN2FBP1ALDH1A1HPGDMAPT
SCHEMBL30905076 0.72 SMN1; SMN2 (0.57) SMN1; SMN2FBP1POLBALDH1A1HPGD
SCHEMBL173265 0.67 FBP1 (1.00) SMN1; SMN2FBP1GAAALDH1A1MEN1
SCHEMBL23122641 0.66 KDM4E (0.46) SMN1; SMN2GAAALDH1A1HPGDMAPT
SCHEMBL7797253 0.65 TXN (0.51) SMN1; SMN2FBP1
SCHEMBL295296 0.65 GAA (0.46) SMN1; SMN2POLBGAAALDH1A1HPGD
SCHEMBL11669798 0.65 GAA (0.46) SMN1; SMN2POLBGAAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2316834-A1 Thiadiazoles or oxadiazoles and their use as inhibitors of JAK protein kinase Vertex Pharmaceuticals Incorporated (US) 2011-05-04 EP disclosed
US-7271179-B2 Inhibitors of JAK protein kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-09-18 US disclosed
US-7271179-B2 Inhibitors of JAK protein kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-09-18 US disclosed
US-4001203-A Heavy metal complexes of azo dyestuffs containing a heterocyclic diazo component and the residue of 5-halogeno-2,3-dihydrozypyridine as coupling component CIBA-GEIGY AG (CH) 1977-01-04 US disclosed