SCHEMBL11706396

SCHEMBL11706396

Cc1cnc2ccc(N3C(=O)c4ccccc4C3=O)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 2/20 0.41
NR1H3 Q13133 2/20 0.39
NPC1 O15118 2/20 0.39
GRM5 P41594 1/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
STAT3 P40763 1/20 0.39
STAT1 P42224 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
MEN1 O00255 1/20 0.39
NR1H2 P55055 1/20 0.38
AR P10275 1/20 0.38
GRM1 Q13255 1/20 0.38
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11484520 0.83 KDM4E (0.39) RAB9ASMN1; SMN2MAPTNR1H3NPC1
SCHEMBL11709729 0.83 NPC1 (0.44) CYP1A2MAPTKMT2ANPC1TP53
SCHEMBL11488725 0.83 NPC1 (0.47) SMN1; SMN2MAPTKMT2ANPC1GRM5
SCHEMBL11709204 0.82 TP53 (0.45) CYP1A2RAB9ASMN1; SMN2MAPTKMT2A
SCHEMBL11709818 0.80 NR1H3 (0.42) NR1H3GRM5KDM4EALDH1A1GAA
SCHEMBL1922080 0.77 SMN1; SMN2 (0.56) RAB9ASMN1; SMN2KMT2ANPC1TP53
SCHEMBL11705831 0.76 ALDH1A1 (0.50) RAB9ASMN1; SMN2MAPTKMT2ATP53
SCHEMBL11608858 0.72 NPC1 (0.54) SMN1; SMN2MAPTKMT2ANPC1KDM4E
SCHEMBL11548784 0.72 HTR1A (0.51) CYP1A2RAB9ASMN1; SMN2MAPTKMT2A
SCHEMBL30046397 0.72 HTR1A (0.51) CYP1A2RAB9ASMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4038391-A TRANQUILIZERS, ANTICONVULSANTS RHONE-POULENC S.A. (FR) 1977-07-26 US disclosed
US-4016274-A TRANQUILIZERS AND ANTICONVULSANT AGENTS RHONE-POULENC S.A. (FR) 1977-04-05 US disclosed