SCHEMBL11709136

SCHEMBL11709136

O=[N+]([O-])Nc1cc(Br)ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
RIOK2 Q9BVS4 1/20 0.38
NTRK1 P04629 1/20 0.34
EGFR P00533 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
IGF1R P08069 2/20 0.33
MITF O75030 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
ERBB2 P04626 1/20 0.33
PTK6 Q13882 1/20 0.33
SORT1 Q99523 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098220 0.78 ALDH1A1 (0.50) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL1897762 0.78 GRM4 (0.38) ALDH1A1RIOK2LMNAMAPTPIK3CA
SCHEMBL27947542 0.74 PKM (0.45) KDM4ERIOK2MAPTHPGDMEN1
SCHEMBL20772265 0.72 MAPT (0.34) SMN1; SMN2NPC1RAB9ALMNAMAPT
SCHEMBL3614808 0.71 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2EGFRIGF1R
SCHEMBL2413590 0.71 NPC1 (0.50) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL31011779 0.71 NPC1 (0.50) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL30413609 0.71 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2EGFRIGF1R
SCHEMBL16913953 0.71 MAPT (0.37) ALDH1A1KDM4ESMN1; SMN2EGFRNPC1
SCHEMBL8501065 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103435561-B A kind of Novel D-amino acid oxidase inhibitor and preparation thereof and application 上海交通大学 2016-08-10 CN disclosed
CN-103435561-A Novel D-amino acid oxidase inhibitor and preparation and application thereof UNIV SHANGHAI JIAOTONG 2013-12-11 CN disclosed
US-4022897-A 4H-PYRIDO(1,2-A) PYRIMIDIN-4-ONE DERIVATIVES E. R. SQUIBB & SONS, INC. (US) 1977-05-10 US disclosed