SCHEMBL11715544

SCHEMBL11715544

COc1cc2c(cc1OC)C(c1ccccc1)N(C(=O)Cl)C(C)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.56
ALDH1A1 P00352 3/20 0.54
LMNA P02545 2/20 0.54
NPC1 O15118 2/20 0.54
MITF O75030 1/20 0.54
XBP1 P17861 1/20 0.54
HTT P42858 1/20 0.54
RAB9A P51151 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
CA14 Q9ULX7 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CA12 O43570 1/20 0.45
CA7 P43166 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11717987 0.77 TRPV1 (0.82) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL22457576 0.75 LMNA (0.50) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL22458078 0.72 ALDH1A1 (0.49) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL22457874 0.72 ALDH1A1 (0.49) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL27542552 0.71 ALDH1A1 (0.46) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL13754594 0.71 TRPV1 (0.84) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL5462519 0.70 TRPV1 (0.82) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL11708173 0.70 ALDH1A1 (0.68) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL11714435 0.70 ALDH1A1 (0.68) TRPV1ALDH1A1LMNANPC1MITF
SCHEMBL9590875 0.70 ALDH1A1 (1.00) TRPV1ALDH1A1LMNANPC1MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4001244-A 1-ARYL-3,4-DIHYDRO-2(1H)-ISOQUINOLINE CARBONYL CHLORIDES G. D. SEARLE & CO. (US) 1977-01-04 US claimed
US-4001244-A 1-ARYL-3,4-DIHYDRO-2(1H)-ISOQUINOLINE CARBONYL CHLORIDES G. D. SEARLE & CO. (US) 1977-01-04 US disclosed