SCHEMBL11729232

SCHEMBL11729232

C[C@H]1Cc2ccccc2[C@H]2CNCC(=O)N21

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.41
HTR2C P28335 10/20 0.41
HTR2A P28223 9/20 0.41
HTR2B P41595 9/20 0.41
PRCP P42785 1/20 0.38
OPRM1 P35372 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11726212 1.00 TAAR1 (0.41) TAAR1HTR2CHTR2AHTR2BPRCP
SCHEMBL30124965 0.78 SRD5A1 (0.42) PRCPOPRM1
SCHEMBL17776282 0.71 TAAR1 (0.54) TAAR1HTR2CHTR2AHTR2B
SCHEMBL14656860 0.71 TAAR1 (0.54) TAAR1HTR2CHTR2AHTR2B
SCHEMBL16019913 0.71 TAAR1 (0.54) TAAR1HTR2CHTR2AHTR2B
SCHEMBL695919 0.71 TAAR1 (0.54) TAAR1HTR2CHTR2AHTR2B
SCHEMBL10484131 0.69 TAAR1 (0.48) TAAR1HTR2CHTR2AHTR2BOPRM1
Phosphoric Acid SCHEMBL31735868 0.66 TAAR1 (0.48) TAAR1HTR2CHTR2AHTR2B
SCHEMBL15468300 0.66 OPRM1 (0.43) OPRM1
SCHEMBL29981061 0.65 HTR2C (0.43) TAAR1HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4049659-A Process for the preparation of 4-oxo-hexahydro-pyrazinoisoquinoline derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-20 US disclosed