SCHEMBL11731998

SCHEMBL11731998

CCOc1ccc2c(c1)C(=O)N(CCCN(C)CCCN1C(=O)c3ccccc3C(C)(C)C1=O)C(=O)C2(C)C

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.48
CYP3A4 P08684 2/20 0.42
MAOB P27338 4/20 0.41
CYP1A2 P05177 1/20 0.41
TSHR P16473 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA1A P35348 1/20 0.41
PGR P06401 1/20 0.40
PDK2 Q15119 1/20 0.40
ALDH1A1 P00352 3/20 0.39
ALOX15 P16050 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RPS6KA2 Q15349 1/20 0.38
ACHE P22303 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11735706 0.88 TDP1 (0.59) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11735486 0.88 TDP1 (0.59) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11734596 0.86 MAOB (0.53) CYP3A4MAOBCYP1A2TSHRADRA2B
SCHEMBL11738968 0.83 TDP1 (0.64) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11738541 0.83 MAOB (0.44) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11734295 0.82 TDP1 (0.58) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11639312 0.79 KMT2A (0.57) CYP3A4MAOBCYP1A2TSHRADRA2B
SCHEMBL11737697 0.78 MAOB (0.51) TDP1CYP3A4MAOBCYP1A2TSHR
SCHEMBL11729888 0.77 MAOB (0.40) TDP1MAOBALOX15MAPTACHE
SCHEMBL11738163 0.77 TDP1 (0.63) TDP1CYP3A4MAOBCYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031219-A ANTIARRHYTHYMICS BOEHRINGER INGELHEIM GMBH (DT) 1977-06-21 US disclosed