SCHEMBL11735486

SCHEMBL11735486

COc1ccc2c(c1)C(=O)N(CCN(C)CCCN1C(=O)c3ccccc3C(C)(C)C1=O)C(=O)C2(C)C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.59
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 2/20 0.48
ALOX15 P16050 1/20 0.48
PGR P06401 1/20 0.47
CYP3A4 P08684 2/20 0.46
CYP1A2 P05177 1/20 0.46
TSHR P16473 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA1A P35348 1/20 0.46
MAOB P27338 5/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
NR1I2 O75469 1/20 0.41
ABCB11 O95342 1/20 0.41
LMNA P02545 1/20 0.41
NR3C1 P04150 1/20 0.41
RARA P10276 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11735706 1.00 TDP1 (0.59) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11738968 0.96 TDP1 (0.64) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11734295 0.95 TDP1 (0.58) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11738163 0.90 TDP1 (0.63) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11731998 0.88 TDP1 (0.48) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11738204 0.86 TDP1 (0.58) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11734596 0.86 MAOB (0.53) PGRCYP3A4CYP1A2TSHRADRA2B
SCHEMBL11737033 0.84 TDP1 (0.56) TDP1KDM4EALDH1A1ALOX15PGR
SCHEMBL11737697 0.83 MAOB (0.51) TDP1PGRCYP3A4CYP1A2TSHR
SCHEMBL11738541 0.83 MAOB (0.44) TDP1PGRCYP3A4CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031219-A ANTIARRHYTHYMICS BOEHRINGER INGELHEIM GMBH (DT) 1977-06-21 US disclosed