SCHEMBL11740137

SCHEMBL11740137

CCOC(=O)c1ccc(OCc2ccccc2)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 7/20 0.57
HPGD P15428 5/20 0.53
RXRA P19793 2/20 0.53
RXRB P28702 2/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
KDM4E B2RXH2 1/20 0.53
RXRG P48443 1/20 0.52
PPIA P62937 2/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
MITF O75030 1/20 0.50
TP53 P04637 1/20 0.50
XBP1 P17861 1/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
ALDH1A1 P00352 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410519 0.93 MRGPRX4 (0.58) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL16584995 0.91 MRGPRX4 (0.58) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL4403626 0.88 SMN1; SMN2 (0.61) MRGPRX4HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL9574663 0.87 MRGPRX4 (0.60) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL3231604 0.86 MRGPRX4 (0.63) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL13440181 0.86 FFAR4 (0.58) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL1561028 0.85 EGFR (0.59) HPGDSMN1; SMN2NPC1RAB9APPIA
SCHEMBL4279981 0.85 HSD17B10 (0.61) MRGPRX4HPGDSMN1; SMN2NPC1RAB9A
SCHEMBL3178525 0.85 HPGD (0.53) MRGPRX4HPGDRXRARXRBSMN1; SMN2
SCHEMBL6508891 0.84 LMNA (0.56) SMN1; SMN2NPC1RAB9AKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4046909-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1977-09-06 US disclosed
US-3998958-A Pyrrolidylidene, piperidylidene and hexahydroazepinylidene ureas as CNS depressants MCNEIL LABORATORIES, INCORPORATED (US) 1976-12-21 US disclosed