SCHEMBL11755459

SCHEMBL11755459

CCc1nsnc1OC[C@@H](O)CNC(C)C

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.46
ADRB1 P08588 4/20 0.46
ADRB3 P13945 2/20 0.46
CYP2D6 P10635 1/20 0.46
PTGS1 P23219 1/20 0.44
SLC6A2 P23975 1/20 0.44
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11755467 1.00 ADRB2 (0.46) ADRB2ADRB1ADRB3CYP2D6PTGS1
SCHEMBL11753904 0.85 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6PTGS1
SCHEMBL11753911 0.85 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6PTGS1
SCHEMBL11411641 0.82 MAPT (0.51) ADRB2ADRB1ADRB3CYP2D6PTGS1
SCHEMBL9749846 0.82 ADRB2 (0.43) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL11753865 0.82 CYP2D6 (0.57) ADRB2ADRB1ADRB3CYP2D6MAPT
SCHEMBL11753852 0.82 CYP2D6 (0.57) ADRB2ADRB1ADRB3CYP2D6MAPT
SCHEMBL9749331 0.81 ADRB2 (0.40) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL11404357 0.81 ADRB2 (0.47) ADRB2ADRB1ADRB3CYP2D6PTGS1
SCHEMBL11754064 0.81 ADRB2 (0.47) ADRB2ADRB1ADRB3CYP2D6PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031125-A 3-Sulfonate ester of 2,3-dihydroxypropylamine MERCK & CO., INC. (US) 1977-06-21 US disclosed
US-3962338-A Novel methods and compounds employed therein MERCK & CO., INC. (US) 1976-06-08 US disclosed