SCHEMBL9749846

SCHEMBL9749846

CC(C)NCC(O)COc1nsnc1CCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.43
ADRB1 P08588 7/20 0.43
ADRB3 P13945 4/20 0.43
CYP2D6 P10635 2/20 0.43
TDP1 Q9NUW8 2/20 0.40
OPRK1 P41145 1/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
PMP22 Q01453 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.39
CNR1 P21554 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749867 0.89 ADRB2 (0.56) ADRB2ADRB1ADRB3CYP2D6TDP1
SCHEMBL9749339 0.86 ADRB2 (0.45) ADRB2ADRB1ADRB3
SCHEMBL9749902 0.84 SMN1; SMN2 (0.52) ADRB2ADRB1ADRB3CYP2D6TDP1
SCHEMBL11755467 0.82 ADRB2 (0.46) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL11755459 0.82 ADRB2 (0.46) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL9749331 0.80 ADRB2 (0.40) ADRB2ADRB1ADRB3CYP2D6TDP1
SCHEMBL11753911 0.79 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL11753904 0.79 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL10994091 0.78 ADRB2 (0.43) ADRB2ADRB1ADRB3CYP2D6TDP1
SCHEMBL9749874 0.76 SMN1; SMN2 (0.34) ADRB2ADRB1ADRB3CYP2D6TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0131006-B1 ESTERS OF 3-(3-SUBSTITUTED-AMINO-2-HYDROXYPROPOXY)-4-SUBSTITUTED-1,2,5-THIADIAZOLE DERIVATIVES THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-06-10 EP claimed