SCHEMBL117564

SCHEMBL117564

NOB(O)c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 1/20 0.38
F3 P13726 1/20 0.38
SARM1 Q6SZW1 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT6 Q8N6T7 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
SIRT4 Q9Y6E7 1/20 0.38
NAPRT Q6XQN6 1/20 0.38
ALDH1A1 P00352 5/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2A6 P11509 3/20 0.38
CYP1A2 P05177 2/20 0.38
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
APP P05067 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8131766 0.83 ALDH1A1 (0.41) F7F3SARM1SIRT2SIRT6
SCHEMBL13712395 0.82 F7 (0.39) F7F3SARM1SIRT2SIRT6
SCHEMBL8515494 0.80 NAPRT (0.38) F7F3SARM1SIRT2SIRT6
SCHEMBL1977767 0.80 CYP2A6 (0.40) F7F3SARM1SIRT2SIRT6
SCHEMBL28011360 0.80 NAPRT (0.38) F7F3SARM1SIRT2SIRT6
SCHEMBL2270306 0.80 ALDH1A1 (0.43) NAPRTALDH1A1CYP3A4CYP2A6CYP1A2
SCHEMBL568870 0.77 ALDH1A1 (0.41) NAPRTALDH1A1CYP3A4CYP2A6CYP1A2
SCHEMBL19737094 0.77
SCHEMBL29376605 0.76
SCHEMBL4647 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424865-A2 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010127237-A2 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed