SCHEMBL11764971

SCHEMBL11764971

C#CC1=C(C)C(=Cc2ccc(Br)cc2)c2ccc(Cl)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 1/20 0.38
PPARG P37231 4/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
RECQL P46063 1/20 0.34
RAB9A P51151 1/20 0.34
MDM2 Q00987 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
RXRA P19793 2/20 0.33
LRRK2 Q5S007 6/20 0.33
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33
APH1A Q96BI3 2/20 0.33
PSENEN Q9NZ42 2/20 0.33
SIRT5 Q9NXA8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11760500 0.92 AMY1A (0.38) AMY1APPARGKDM4EPOLBMAPT
SCHEMBL11765128 0.92 PPARG (0.37) PPARGKDM4EPOLBMAPTRECQL
SCHEMBL11765459 0.87 PPARG (0.47) PPARGKDM4EMAPTNPSR1TDP1
SCHEMBL11764094 0.86 MAPT (0.36) AMY1APPARGKDM4EPOLBMAPT
SCHEMBL11763054 0.85 PSEN1 (0.42) PPARGKDM4EMAPTMDM2RXRA
SCHEMBL11767110 0.84 PPARG (0.50) PPARGKDM4EMAPTNPSR1TDP1
SCHEMBL11765291 0.84 MAPT (0.39) AMY1APPARGKDM4EPOLBMAPT
SCHEMBL11763704 0.84 RXRA (0.47) PPARGMAPTTDP1RXRAPSEN1
SCHEMBL11764221 0.83 LRRK2 (0.33) PPARGMAPTNPSR1TDP1RXRA
SCHEMBL11765230 0.82 LCK (0.40) PPARGMAPTRXRALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4061771-A Ethynylindenyl compounds and derivatives thereof used in the treatment of pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1977-12-06 US disclosed
US-3983253-A Ethynylindenyl compounds and derivatives thereof used in the treatment of pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1976-09-28 US disclosed