SCHEMBL11786153

SCHEMBL11786153

Nc1ncc(Cl)nc1C(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.55
MAPKAPK2 P49137 4/20 0.48
GLA P06280 1/20 0.44
HPGD P15428 1/20 0.44
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
ATR Q13535 7/20 0.42
PRKDC P78527 2/20 0.42
PIK3CD O00329 1/20 0.42
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30504276 1.00 GRM5 (0.55) GRM5MAPKAPK2GLAHPGDCDK5
SCHEMBL1318334 0.83 GRM5 (0.51) GRM5MAPKAPK2ATRPRKDCALDH1A1
SCHEMBL3408307 0.82 ATR (0.61) GRM5CDK5CDK5R1ATRPRKDC
SCHEMBL3374259 0.81 CDK5 (0.43) GLAHPGDCDK5CDK5R1ATR
SCHEMBL12343678 0.81 GRM5 (0.55) GRM5MAPKAPK2CDK5CDK5R1ATR
SCHEMBL14015128 0.80 HPGD (0.50) GRM5MAPKAPK2GLAHPGDALDH1A1
SCHEMBL5684569 0.79 ATR (0.63) CDK5CDK5R1ATRPRKDC
SCHEMBL11008090 0.78 ALDH1A1 (0.45) GRM5GLAHPGDCDK5CDK5R1
SCHEMBL3860081 0.77 ATR (0.72) GRM5ATRPRKDC
SCHEMBL11263012 0.77 MAPT (0.46) GLAHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3954753-A SEDATIVES, MUSCLE RELAXANTS, ANTICONVULSANTS HOFFMANN-LA ROCHE INC. (US) 1976-05-04 US disclosed