SCHEMBL117977

SCHEMBL117977

Cn1ccnc1-c1cc(C(F)(F)F)ncc1F

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
LRRK2 Q5S007 1/20 0.35
SCN9A Q15858 2/20 0.35
SCN10A Q9Y5Y9 6/20 0.34
ATR Q13535 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
DPP4 P27487 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
LPO P22079 1/20 0.31
HCRTR1 O43613 1/20 0.31
CCNC P24863 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719531 0.85 LRRK2 (0.42) BRD4LRRK2SCN9ANPC1RAB9A
SCHEMBL3728805 0.84 LRRK2 (0.41) BRD4LRRK2SCN9ANPC1RAB9A
SCHEMBL3796268 0.81 LRRK2 (0.40) BRD4LRRK2SCN9A
SCHEMBL3722934 0.81 BRD4 (0.37) BRD4LRRK2SCN9AADRA1DADRA1A
SCHEMBL3722905 0.81 BRD4 (0.37) BRD4LRRK2SCN9ASCN10ANPC1
SCHEMBL3727131 0.79 LRRK2 (0.39) BRD4LRRK2SCN9ANPC1RAB9A
SCHEMBL3723882 0.79 LRRK2 (0.39) BRD4LRRK2SCN9A
SCHEMBL3721949 0.79 SCN9A (0.35) BRD4LRRK2SCN9A
SCHEMBL3721068 0.79 SCN9A (0.36) BRD4LRRK2SCN9A
SCHEMBL3720890 0.79 LRRK2 (0.41) BRD4LRRK2SCN9ASCN10AHCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424856-A1 FUSED HETEROCYCLIC COMPOUND AND USE THEREOF Sumitomo Chemical Company, Limited (JP) 2012-03-07 EP disclosed
WO-2010125985-A1 FUSED HETEROCYCLIC COMPOUND AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-11-04 WO disclosed