SCHEMBL3722934

SCHEMBL3722934

CSc1cnc(C(F)(F)F)cc1-c1nccn1C

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SCN9A Q15858 2/20 0.34
LRRK2 Q5S007 1/20 0.34
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
BDKRB2 P30411 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721717 0.85 NPC1 (0.37) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL3719531 0.81 LRRK2 (0.42) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL117977 0.81 BRD4 (0.36) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL3728805 0.80 LRRK2 (0.41) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL3722905 0.78 BRD4 (0.37) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL3796268 0.78 LRRK2 (0.40) BRD4SCN9ALRRK2BDKRB2
SCHEMBL3721068 0.76 SCN9A (0.36) BRD4SCN9ALRRK2
SCHEMBL3723882 0.76 LRRK2 (0.39) BRD4SCN9ALRRK2BDKRB2KDM4E
SCHEMBL3727131 0.76 LRRK2 (0.39) BRD4NPC1RAB9ASCN9ALRRK2
SCHEMBL3721949 0.76 SCN9A (0.35) BRD4SCN9ALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125985-A1 FUSED HETEROCYCLIC COMPOUND AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-11-04 WO disclosed