SCHEMBL11802486

SCHEMBL11802486

C#Cc1ccc(Oc2ccccc2)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 1/20 0.44
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
HAO1 Q9UJM8 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNE1 P15382 1/20 0.37
KCNQ1 P51787 1/20 0.37
LTA4H P09960 1/20 0.37
TSHR P16473 1/20 0.37
TTR P02766 1/20 0.37
HSPB1 P04792 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11794954 0.84 HSPB1 (0.42) SLC6A4HAO1HSPB1
SCHEMBL923176 0.83 ERBB2 (0.53) ERBB2HTR2ASLC6A4
SCHEMBL25532058 0.82 HSPB1 (0.37) ERBB2HSPB1
SCHEMBL25532070 0.82 HSPB1 (0.37) ERBB2HTR2ASLC6A4HSPB1
SCHEMBL432736 0.82 SMN1; SMN2 (0.52)
SCHEMBL25532060 0.80 L3MBTL1 (0.36) HTR2ASLC6A4HAO1HSPB1
SCHEMBL25532048 0.80 MAPT (0.36) HTR2ASLC6A4CYP1A2TSHRHSPB1
SCHEMBL11311431 0.79 NTRK1 (0.43) CYP1A2CYP3A4CYP2C9CYP2C19LTA4H
SCHEMBL11792502 0.79 HSPB1 (0.54) HTR2ASLC6A4HSPB1
SCHEMBL25532053 0.79 KDM4E (0.38) ERBB2HSPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3939278-A Phenoxyphenyl-acetylenes and thio analogues thereof as antithrombotic agents ELI LILLY AND COMPANY (US) 1976-02-17 US disclosed