SCHEMBL11804792

SCHEMBL11804792

COC(=O)CN1C(=O)CN=C(c2c(F)cccc2F)c2cc(Cl)ccc21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.58
MAPT P10636 4/20 0.54
OPRK1 P41145 3/20 0.53
KCNH2 Q12809 2/20 0.53
HTR1A P08908 1/20 0.53
DRD3 P35462 1/20 0.53
HTR3A P46098 1/20 0.53
GHSR Q92847 1/20 0.53
NPSR1 Q6W5P4 2/20 0.53
ALDH1A1 P00352 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CYP1A2 P05177 1/20 0.52
MCL1 Q07820 1/20 0.51
GABRP O00591 2/20 0.50
GABRD O14764 2/20 0.50
GABRA1 P14867 2/20 0.50
GABRB1 P18505 2/20 0.50
GABRG2 P18507 2/20 0.50
GABRB3 P28472 2/20 0.50
GABRA5 P31644 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11805034 0.89 TP53 (0.47) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL11806947 0.85 MAPT (0.72) TP53MAPTOPRK1KCNH2NPSR1
SCHEMBL11802020 0.84 MAPT (0.65) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL11802793 0.80 TP53 (0.46) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL11811476 0.80 TP53 (0.55) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL11812864 0.78 RAB9A (0.57) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL9727938 0.78 CYP1A2 (0.70) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL11812609 0.77 TP53 (0.52) TP53MAPTOPRK1KCNH2HTR1A
SCHEMBL5352101 0.75 NPSR1 (0.69) TP53MAPTOPRK1KCNH2NPSR1
SCHEMBL9038774 0.74 NPSR1 (0.65) TP53MAPTOPRK1KCNH2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3933816-A 3-(Substituted aminomethyl)-7-substituted-3,5-dihydro-as-triazino[4,3-a][1,5]benzodiazepines THE UPJOHN COMPANY (US) 1976-01-20 US disclosed