SCHEMBL11821663

SCHEMBL11821663

C=CC(C#N)c1cccc(C)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 2/20 0.38
HTT P42858 1/20 0.38
CCR1 P32246 1/20 0.36
CCR8 P51685 1/20 0.36
NOS3 P29474 1/20 0.34
NOS2 P35228 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.32
GRM5 P41594 4/20 0.32
ALDH1A1 P00352 3/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
HDAC6 Q9UBN7 2/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C9 P11712 2/20 0.32
PKM P14618 2/20 0.32
HPGD P15428 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3524973 0.76 L3MBTL1 (0.46) RECQLHTTCCR1CCR8NOS3
SCHEMBL11826583 0.73 HTT (0.41) RECQLHTTCCR1CCR8NOS3
SCHEMBL11822739 0.73 HTT (0.41) RECQLHTTCCR1CCR8NOS3
SCHEMBL4558714 0.71 SMN1; SMN2 (0.42) ALDH1A1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL11814736 0.70 HTT (0.39) RECQLHTTCCR1CCR8NOS3
SCHEMBL11631991 0.69 L3MBTL1 (0.51) RECQLHTTGRM5ALDH1A1NPC1
SCHEMBL954513 0.68 CCR1 (0.52) RECQLHTTCCR1CCR8NOS3
SCHEMBL16545967 0.68 HTT (0.37) RECQLHTTCCR1CCR8NOS3
SCHEMBL17331400 0.68 HTT (0.37) RECQLHTTCCR1CCR8NOS3
SCHEMBL1706922 0.67 CCR1 (0.46) RECQLHTTCCR1CCR8NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3950522-A N-ALKENYL OR N-ALKYNYL THIOAMIDES SMITHKLINE CORPORATION (US) 1976-04-13 US disclosed
US-3932641-A THIOACETAMIDES SMITHKLINE CORPORATION (US) 1976-01-13 US disclosed
US-3931162-A N-Aminomethyl heterocyclic thioacetamides SMITHKLINE CORPORATION (US) 1976-01-06 US disclosed